antagonists and inhibitors
Rev. esc. enferm. USP vol.49 número1
... channel antagonists and inhibitors of angiotensin-converting enzyme in plasma concentrations of hydrogen sulide and nitric oxide in patients with ...enzyme inhibitors or calcium channel ...
6
Effects of α-adrenoceptor antagonists on ABCG2/BCRP-mediated resistance and transport.
... resistance, and remains a critical factor in the success of cancer ...the inhibitors for multidrug ...a-adrenoceptor antagonists on ABCG2/BCRP-mediated resistance and ...the antagonists ...
8
Human fetal malformations associated with the use of an angiotensin II receptor antagonist: Case Report
... obstetrics and data regarding the safety of antihypertensive drugs during pregnancy are relatively ...weeks and 4 days of gestation. She reported a history of hypertension and was currently being ...
4
Arq. Gastroenterol. vol.54 número4
... infant))) AND ((((Histamine H2 Antagonists OR ranitidine OR ranitidine OR cimetidine))) OR ((Proton Pump Inhibitors OR omeprazole OR pantoprazole OR lansoprazole OR esomeprazole OR rabeprazole)))) ...
10
CAFFEOYLQUINIC ACIDS AND THEIR METABOLITES AS INHIBITORS FOR ALFA- GLUCOSIDASE
... bulky and was expected to interact with a lot of residues which was not what resulted from the ...abandoned and the design process focused on starting with smaller ligands and optimizing them to ...
116
Comparison of Inhibitory Activities of <i>meta</i> and <i>para</i> Substituted <i>N</i>-aryl 3-Hydroxypyridin-4-one Mannosides Towards Type 1 Fimbriated <i>E. coli</i>
... Reagents and solvents for the synthesis of compounds were obtained from commercial sources (Sigma-Aldrich ...Corp. and J. T. Baker). When necessary solvents were further purified and/or dried using ...
6
Cholinesterase inhibitors and hospitalization for bradycardia: a population-based study.
... cholinesterase inhibitors increase the risk of bradycardia, an abnormally slow resting heart rate of below 60 beats a minute, which can cause fatigue, dizziness, fainting, palpitations, shortness of breath, or ...
9
The Interaction of Clopidogrel and Proton Pump Inhibitors
... clopidogrel and proton pump inhibitors following acute coronary ...therapy and NSAID use: a report of the American College of Cardiology Foundation Task Force on Clinical Consensus ...
3
Expression, Purification and Activity Assay of Two New Recombinant Antagonists of Fibrinogen Receptor
... disease and stroke, have proven to be closely related with ...world and badly hurt the health of human beings [1] ...receptor and is a potent inhibitor of platelet ...long and contains 6 ...
5
Arq. Gastroenterol. vol.49 número4
... The development of investigative tests, such as the study of relux by impedance/pH-metry, high-resolution esopha- geal manometry and gastric scintigraphy will probably con- tribute to better identify GERD. Such ...
6
Arq Bras Endocrinol Metab vol.49 número5
... tumor and hepatic metastasis ...Williams and Sandler classified carcinoids according to their embryologic site of origin as foregut carcinoids (respiratory tract, stomach, duodenum, biliary system, ...
11
Effectiveness inactivation of trypsin inhibitor fron brazilian cultivarof beans (Phaseolus vulgaris L.)
... raw and pressure-cooking IAC-Aruã beans have showed similar hydrolysis degree by pepsin at least for 180 minutes (Figure 1), the pressure-cooking at 121ºC for 30 min increased the susceptible to proteolysis by ...
7
TRIB2 confers resistance to MAPK and TOR1 inhibitors
... contacts and cell-matrix interactions (integrins and cadherins) or through the action of secreted signalling ...paracrine and autocrine ...cells and in autocrine signalling, a cell produces a ...
96
Discovery and computer aided potency optimization of a novel class of small molecule CXCR4 antagonists.
... blood and breast ...CXCR4 antagonists based on the use of computational modelling studies in concert with experimental determination of in vitro activity against CXCL12-induced intracellular calcium ...
18
Rev. Soc. Bras. Med. Trop. vol.50 número5
... enteritis and Crohn’s ...age and had received oral prednisolone and oral and subcutaneous methotrexate for a period of 3 ...etanercept and prednisolone for 7 ...fever and ...
3
Montelukast reduces seizures in pentylenetetrazol-kindled mice
... group and other studies indicating that systemic montelukast does not prevent PTZ-induced seizures in mice, as well as evidence that montelukast and pranlukast cross the BBB ...
7
Efficacy and mode of action of yeast antagonists for control of Penicillium digitatum in oranges
... as antagonists is due in part to their ability to rapidly colonize wound sites despite low nutrient ...of antagonists lyse pathogen hyphae and thereby increase the availability of simple carbon ...
8
Nanoscale Synaptic Membrane Mimetic Allows Unbiased High Throughput Screen That Targets Binding Sites for Alzheimer's-Associated Aβ Oligomers.
... enzymatic and ligand binding activity consistent with conformational ...affinity and specificity, with binding dependent on intact synaptic membrane proteins, and selective for the higher molecular ...
24
J. Braz. Chem. Soc. vol.23 número11
... model and could not be ...plotted and the results are shown in Figure ...model and there is no outlier compound both for training and test sets, indicating the reliability of the ...
11
Blockade of Neuronal Facilitatory Nicotinic Receptors Containing
... (Schuetze and Role, 1987; Salpeter et ...Meca, and HEX could simul- taneously depress tetanic peak tension, reduce evoked [ 3 H]-ACh release, and induce tetanic fade, as ...
12