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Biological evaluation

Synthesis, biological evaluation and molecular modeling of arylfurans as potential trypanothione reductase inhibitors.

Synthesis, biological evaluation and molecular modeling of arylfurans as potential trypanothione reductase inhibitors.

... SYNTHESIS, BIOLOGICAL EVALUATION AND MOLECULAR MODELING OF ARYLFURANS AS POTENTIAL TRYPANOTHIONE REDUCTASE INHIBITORS. Trypanosoma cruzi is a protozoan parasite that causes a severe disease (Chagas’disease) ...

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Synthesis and biological evaluation of mono and bis-naphthalimide derivatives against SH-SY5Y, human brain cancer cells

Synthesis and biological evaluation of mono and bis-naphthalimide derivatives against SH-SY5Y, human brain cancer cells

... 26.Banerjee, S.; Veale, E. B.; Phelan, C. M.; Murphy, S. A.; Tocci, G. M.; Gillespie, L. J.; Frimannsson, D. O.; Kelly, J. M.; Gunnlaugsson, T., Recent advances in the development of 1,8-naphthalimide based DNA targeting ...

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BIOLOGICAL EVALUATION OF CHLORELLA RESINOID VIA PARAMECIUM CAUDATUM

BIOLOGICAL EVALUATION OF CHLORELLA RESINOID VIA PARAMECIUM CAUDATUM

... its biological availability and efficiency some other approaches based on complex formations of silver together with ligands and stabilization of silver with polymers were used ...

148

Biological evaluation of recombinant human erythropoietin in pharmaceutical products

Biological evaluation of recombinant human erythropoietin in pharmaceutical products

... the biological activity of rhEPO is measured by the stimulation of reticulocyte production ...potency evaluation of pharmaceutical preparations (13,15,19); however, although they are usually robust, some ...

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Biological evaluation of isoniazid derivatives as an anticancer class

Biological evaluation of isoniazid derivatives as an anticancer class

... A series of thirty-two isoniazid derivatives have been evaluated for their activity against four human cancer cell lines with potent cytotoxicity (IC50 ranging from 0.61 to 3.36 μ g/mL). The structure-activity ...

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Biochemical and biological evaluation of gyroxin isolated from Crotalus durissus terrificus venom

Biochemical and biological evaluation of gyroxin isolated from Crotalus durissus terrificus venom

... Crotalus durissus terriicus snake venom, vacuum dried and stored at 4°C, was obtained from specimens kept in the serpentarium of the Center for the Studies of Venoms and Venomous Animals (CEVAP), São Paulo state, Brazil. ...

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3-Hydroxy-quinolin-2(1H)-ones, a useful scaffold : synthesis and biological evaluation

3-Hydroxy-quinolin-2(1H)-ones, a useful scaffold : synthesis and biological evaluation

... the biological activity of 3HQ and its ...important biological studies were performed on 4-carboxamide-3HQ derivatives showed interesting biological activity as a potential anticancer lead ...

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Biological Evaluation of Chlorogold Complexes as Potential Anti-Tumoural Compounds: Unraveling Mechanisms of Action

Biological Evaluation of Chlorogold Complexes as Potential Anti-Tumoural Compounds: Unraveling Mechanisms of Action

... 15 morphological alterations already mentioned above (Elmore, 2007). A noteworthy concept to keep in mind is that once activated, cells seemingly become committed to a programmed cell death. At the risk of being over ...

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Synthesis and biological evaluation of novel benzo[b]xanthone derivatives as potential antitumor agents

Synthesis and biological evaluation of novel benzo[b]xanthone derivatives as potential antitumor agents

... and biological activities by the introduction of a nitro- gen-containing side chain 17 and the structure of 1,3-dihydroxybenzoxanthone, in the herein reported study, a series of novel benzo[b]xanthone derivatives ...

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Design synthesis and biological evaluation of new antiplasmodial compounds related to ellagic acid

Design synthesis and biological evaluation of new antiplasmodial compounds related to ellagic acid

... Malaria remains a major public health problem, especially in subtropical regions. This endemic disease is caused by parasitic protozoans that belong to the Plasmodium type and people who get malaria are typically very ...

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Cyclopentenones: synthesis and biological evaluation in human cancer cells

Cyclopentenones: synthesis and biological evaluation in human cancer cells

... From ancient times, human beings strive to discover the cure of diseases that affect them. Before the twentieth century, they used to treat diseases by rudimentary techniques such the use of medicinal herbs and potions, ...

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Synthesis and biological evaluation of novel 6Hydroxybenzo[d]oxathiol2one Schiff bases as potential anticancer agents

Synthesis and biological evaluation of novel 6Hydroxybenzo[d]oxathiol2one Schiff bases as potential anticancer agents

... In this context, several heterocyclic systems with five-membered rings fused to a benzene nucleus play an important role on designing of new drugs, since they display an interesting and diversified pharmacological ...

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SYNTHESIS OF SULFONAMIDE BASED SCHIFF’S BASES AND THEIR BIOLOGICAL EVALUATION TOWARDS COLLETOTRICHUM GLOEOSPORIOIDES

SYNTHESIS OF SULFONAMIDE BASED SCHIFF’S BASES AND THEIR BIOLOGICAL EVALUATION TOWARDS COLLETOTRICHUM GLOEOSPORIOIDES

... of biological activities and industrial ...various biological and pharmacological ...several biological application 15-16 ...and biological activities 17-19 ...

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Rev. bras. farmacogn.  vol.26 número1

Rev. bras. farmacogn. vol.26 número1

... the biological and toxicological potential of this ...The biological evaluation was performed by the determination of cyto- toxic (MTT and hemolysis assay) and immunomodulatory (phagocytic capacity, ...

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Anti-inflammatory drug design by molecular hybridization approach

Anti-inflammatory drug design by molecular hybridization approach

... Dinitroglyceryl and diazen-1-ium-1,2-diolated nitric oxide donor ester prodrugs of aspirin, indomethacin and ibuprofen: Synthesis, biological evaluation and nitric oxide release studie[r] ...

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Rev. bras. farmacogn.  vol.17 número4

Rev. bras. farmacogn. vol.17 número4

... Following ecdysis, fi fth-instar nymphae of male R. prolixus were starved for 25 days. Insects were then submitted to three different approaches. In the control group I insects were only fully engorged on citrated whole ...

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J. Braz. Chem. Soc.  vol.25 número10

J. Braz. Chem. Soc. vol.25 número10

... and biological evaluation (TcTS inhibition and antitrypanosomal activities) of some galactose-containing triazol-arylsulfonamides via microwave-assisted Cu(I) 1,3-dipolar azide-alkyne cycloaddition (CuAAC) ...

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Synthesis and antitubercular evaluation of new 1,2,3-triazole derivatives of carbohydrates

Synthesis and antitubercular evaluation of new 1,2,3-triazole derivatives of carbohydrates

... several biological activities including antibacterial, herbicidal, fungicidal, antiallergic and anti-HIV 2,3 ...and biological evaluation of their glicoconjugates, have been shown to stand out as HIV ...

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Nonspecific blockade of vascular free radical signals by methylated arginine analogues

Nonspecific blockade of vascular free radical signals by methylated arginine analogues

... Our data, as well as the observations discussed above, underscore the importance of adequate controls for the evaluation of the biological roles of nitric oxide. On the basis of these data, we propose that ...

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Biocontrol agents in the management of Meloidogyne incognita in tomato

Biocontrol agents in the management of Meloidogyne incognita in tomato

... the biological control of nematodes, especially the root-knot nematodes, as it is a fungus that parasitizes females and eggs, the later being the most vulnerable stage of this pathogen life ...

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