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[PDF] Top 20 Synthesis and antitubercular evaluation of new 1,2,3-triazole derivatives of carbohydrates

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Synthesis and antitubercular evaluation of new 1,2,3-triazole derivatives of carbohydrates

Synthesis and antitubercular evaluation of new 1,2,3-triazole derivatives of carbohydrates

... preparation of novel 1,4-disubstituted-1,2,3-triazoles derivatives from D- glucose and D-fructose and their in vitro antibacterial activity against Mycobacterium tuberculosis were ...chemical ... See full document

7

Synthesis and evaluation of antimalarial activity of curcumin derivatives.

Synthesis and evaluation of antimalarial activity of curcumin derivatives.

... SYNTHESIS AND EVALUATION OF ANTIMALARIAL ACTIVITY OF CURCUMIN ...One of the main challenges in the development of new antimalarial drugs is to achieve a viable lead ... See full document

5

Synthesis and Anti-Mycobacterium tuberculosis Evaluation of Aza-Stilbene Derivatives

Synthesis and Anti-Mycobacterium tuberculosis Evaluation of Aza-Stilbene Derivatives

... one of the leading causes of death in the world, reaching a million deaths ...2007 and 456,000 deaths among individuals infected with both TB and ...TB, and TB/HIV are stifling attempts ... See full document

8

Synthesis and antimicrobial activity of new amino derivatives of pyrano[4’’,3’’:4’,5’]pyrido[3’,2’:4,5]thieno[3,2-d]pyrimidine

Synthesis and antimicrobial activity of new amino derivatives of pyrano[4’’,3’’:4’,5’]pyrido[3’,2’:4,5]thieno[3,2-d]pyrimidine

... pyridine-2-carboxylate 1 (Sirakanyan et al. 2014) was used. Compound 1 reacts with benzoyl isothiocyanate in benzene, giving the relevant thioureido derivative 2, which in turn underwent ... See full document

15

Synthesis and Antibacterial Evaluation of 3,5-Diaryl-1,2,4-oxadiazole Derivatives

Synthesis and Antibacterial Evaluation of 3,5-Diaryl-1,2,4-oxadiazole Derivatives

... the synthesis of twenty 3,5-diaryl-1,2,4-oxadiazole derivatives, nine of which are novel ...mirabilis and Staphylococcus ...(MIC) of the active compounds were determined by ... See full document

12

One pot synthesis of 2-hydroxy pyrrolidine derivatives

One pot synthesis of 2-hydroxy pyrrolidine derivatives

... utility of domino reaction between aryl amines, in particularly with various anilines and cyclic enol ethers such as 2,3-dihydrofuran and 3,4-dihydro-2H-pyran in the straight forward synthesis ... See full document

6

Synthesis, cytotoxicity and mechanistic evaluation of 4oxoquinoline3carboxamide derivatives : finding new potential Aaticancer drugs

Synthesis, cytotoxicity and mechanistic evaluation of 4oxoquinoline3carboxamide derivatives : finding new potential Aaticancer drugs

... doublet of doublets; t, triplet; q, quartet; m, multiplet. Hydrogen and carbon NMR spectra were typically obtained at room ...pellets, and frequencies were expressed in cm −1 ... See full document

20

J. Braz. Chem. Soc.  vol.23 número6

J. Braz. Chem. Soc. vol.23 número6

... incorporation of a 1,2,3-triazole heterocyclic unit into 3-nitrocoumarins might provide 1,2,3-triazole derivatives that have important biological and pharmaceutical ...possible ... See full document

15

Synthesis and antifungal evaluation of imines derived from 3-Amino-2-isopropyl-3H-quinazolin-4-one

Synthesis and antifungal evaluation of imines derived from 3-Amino-2-isopropyl-3H-quinazolin-4-one

... variety of quinazolinone-based alkaloid natural and non-natural products have been known for their biological properties, for example, antitumor, 1-4 anti-inflammatory, 5-7 anticonvulsant, 8-11 ... See full document

9

Synthesis and evaluation of the phytotoxic activity of α-Santonin derivatives.

Synthesis and evaluation of the phytotoxic activity of α-Santonin derivatives.

... Pentan-3-ona (24 µL), xileno (48 µL), monoleato de polietileno glicol (Tween 80, 72 µL), água destilada (2 mL) e o composto avaliado (0,02 mmol) foram adicionados a um tubo de ensaio. Após este tubo ter ... See full document

6

Design, synthesis and biological evaluation of (E)2(2)quinoxalines, a promising and potent new class of anticancer agents

Design, synthesis and biological evaluation of (E)2(2)quinoxalines, a promising and potent new class of anticancer agents

... thesized and evaluated for their activity against four cancer cell lines: potent cytotoxicities were found (IC 50 ranging from ...positions and the type of substituents attached to the aromatic ring ... See full document

6

Design, synthesis and the effect of 1,2,3-triazole sialylmimetic neoglycoconjugates on Trypanosoma cruzi and its cell surface trans-sialidase

Design, synthesis and the effect of 1,2,3-triazole sialylmimetic neoglycoconjugates on Trypanosoma cruzi and its cell surface trans-sialidase

... triad and Tyr342 at the donor ...their triazole rings and Trp312, while galactosyl moiety of 13 was capable to interact, additionally, with both Trp312 and Tyr119 ...Figure 3, ... See full document

12

SYNTHESIS AND ANTIMICROBIAL ACTIVITIES OF NEW PYRAZOLOPYRIDAZINE DERIVATIVES

SYNTHESIS AND ANTIMICROBIAL ACTIVITIES OF NEW PYRAZOLOPYRIDAZINE DERIVATIVES

... Several new pryrazolo-pyridazine derivatives (4a-h) were synthesized through multi-step synthesis and evaluated for their antimicrobial ...with 2 to furnish pyridazinone ... See full document

7

Synthesis of Triazole Schiff's Base Derivatives and Their Inhibitory Kinetics on Tyrosinase Activity.

Synthesis of Triazole Schiff's Base Derivatives and Their Inhibitory Kinetics on Tyrosinase Activity.

... center of tyrosinase were the central part of catalytic activities of tyrosinase and it were found in the enzyme from different species ...So synthesis and screening of ... See full document

13

Synthesis and antimicrobial activity of new 3,5-diarylidene-4-piperidone derivatives

Synthesis and antimicrobial activity of new 3,5-diarylidene-4-piperidone derivatives

... mixture of 4-piperidone hydrochloride monohydrate (1, 10 mmol) and various substituted aromatic aldehydes (20 mmol) in ethanol (10 mL) was stirred at room temperature (29 °C) for 10 ...progress ... See full document

12

J. Braz. Chem. Soc.  vol.18 número6

J. Braz. Chem. Soc. vol.18 número6

... mass 1-alkyl-4-phenyl-[1,2,3]-triazole derivatives were prepared using a straightforward and efficient method for the regioselective synthesis of [1,2,3]-triazoles and the ... See full document

7

Synthesis and preliminary evaluation of N-oxide derivatives for the prevention of atherothrombotic events

Synthesis and preliminary evaluation of N-oxide derivatives for the prevention of atherothrombotic events

... mg/kg) and negative control (1% carboxymethylcellulose (CMC) suspension and ...Groups of 10 Swiss mice of both sexes (25 −30 g) were used in each test and control ...mixture ... See full document

16

Synthesis of 1,2,3-Triazole Derivatives of 4,4’-Dihydroxybenzophenone and Evaluation of Their Elastase Inhibitory Activity

Synthesis of 1,2,3-Triazole Derivatives of 4,4’-Dihydroxybenzophenone and Evaluation of Their Elastase Inhibitory Activity

... separated and the aqueous layer was extracted with ethyl acetate (3 × 20 ...combined and the resulting organic layer was washed with brine, dried over anhydrous sodium sulfate, and ... See full document

11

J. Braz. Chem. Soc.  vol.28 número4

J. Braz. Chem. Soc. vol.28 número4

... the synthesis of 2-amino-alkyl-1,2,3-triazole-1,4- naphthoquinone derivatives make it possible to obtain desired products from 1,4-naphthoquinone (1,4-NQ), and bio-based lawsone, ... See full document

8

INSTITUTIONS IN TRANSITION: IS THE EU INTEGRATION PROCESS RELEVANT FOR INWARD FDI IN TRANSITION EUROPEAN ECONOMIES?

INSTITUTIONS IN TRANSITION: IS THE EU INTEGRATION PROCESS RELEVANT FOR INWARD FDI IN TRANSITION EUROPEAN ECONOMIES?

... definition of local content policy (LCP) and often different companies and countries employ different measurements for ...‗amount‘ of domestically produced inputs in producing its final ... See full document

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