[PDF] Top 20 Studies on new substituted pyridazinones: synthesis and biological evaluation
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Studies on new substituted pyridazinones: synthesis and biological evaluation
... (MDR-TB) and an ever increasing emergence of extensively drug-resistant (XDR) TB (Asif, ...interfere and inhibit cell processes of growing ...develop new TB drugs having both bactericidal as well as ... See full document
12
Synthesis of new antibiotic glycosides and computational studies on their interaction with model lipid bilayers
... simulated and preliminarily an- alyzed with respect to their relative stabilities and configurations in ...report on the results from a series of simulations performed starting from several ... See full document
209
Synthesis and biological evaluation of novel benzo[b]xanthone derivatives as potential antitumor agents
... 1.59 and 5.47 μМ, respectively. However, for the cell lines BEL- 7402 and MGC-803, compounds 3c and 3d, which have N-heterocyclic rings at the C-3 position of ... See full document
8
SYNTHESIS OF SULFONAMIDE BASED SCHIFF’S BASES AND THEIR BIOLOGICAL EVALUATION TOWARDS COLLETOTRICHUM GLOEOSPORIOIDES
... sulfonamide and substituted aromatic aldehydes were dissolved in minimum amount of ...added and refluxed for about 6-8 hours then cools to room temperature and the content was poured on ... See full document
3
Synthesis and evaluation of new pyrazoles, glycosylpyrazoles and rutheniumpyrazoles for antioxidant and antitumoral activity
... 5.1 and Figure ...depends on the structure and the substitution pattern of the R group in position ...9 and 10 was significantly lower (from ...role on the antioxidant effect, the free ... See full document
88
Design, synthesis and biological evaluation of (E)2(2)quinoxalines, a promising and potent new class of anticancer agents
... thesized and evaluated for their activity against four cancer cell lines: potent cytotoxicities were found (IC 50 ranging from ...positions and the type of substituents attached to the aromatic ring are ... See full document
6
Design, synthesis, biological evaluation, and nitric-oxide release studies of a novel series of celecoxib prodrugs possessing a nitric-oxide donor moiety
... vivo and in vitro studies on NO-aspirin displayed more potent antithrombic properties when compared to ...NO-flurbiprofen and NO-aspirin incapacitated the brain’s inflammatory response ... See full document
10
Macroevolution and macroecology for the biological synthesis
... the biological hierarchies. An example is provided on how the higher levels may constrain and enhance our knowledge of lower level ...Evolutionary Synthesis is appropriate for the organismic ... See full document
8
ARTIGO_Synthesis, biological evaluation and docking studies of novel bisquaternary aldoxime reactivators
... the synthesis and in vitro evaluation of three novel bisquaternary aldoximes as potential reactivators for HssAChE and HssBChE inhibited by the pesticide POX, which failed to reactivate these ... See full document
11
Cyclopentenones: synthesis and biological evaluation in human cancer cells
... working on the preparation of trans-4,5-diaminocyclopentenones from furfural (cheap furan derivative, easily available and obtained from non-edible carbohydrates such as ...CP and was also observed ... See full document
132
New Fully Biodegradable PEG-Dendrimers: Synthesis and evaluation as siRNA vectors
... vitro and in vivo results in several research labs around the world, not so many have gone into clinical trials, especially due to their ...effect on cells is mainly caused by bioaccumulation and, ... See full document
80
3-Hydroxy-quinolin-2(1H)-ones, a useful scaffold : synthesis and biological evaluation
... natural and synthetic molecules and a broad spectrum of biological properties like, antimicrobial, enzymatic and neuro protective activities, have been attributed to these ...(4HQs) and ... See full document
233
Synthesis, biological evaluation and molecular modeling of arylfurans as potential trypanothione reductase inhibitors.
... SYNTHESIS, BIOLOGICAL EVALUATION AND MOLECULAR MODELING OF ARYLFURANS AS POTENTIAL TRYPANOTHIONE REDUCTASE ...Central and South ...of new drugs against this ...based on ... See full document
7
Synthesis of new sugar derivatives containing an α, β-unsaturated carbonyl system in their structure and biological evaluation
... alditols and aldoses catalyzed by a transition metal complex in the presence of a hydrogen acceptor ...the synthesis of aldonolactones/aldonic acids are preferred on industrial ... See full document
293
Synthesis and antitubercular evaluation of new 1,2,3-triazole derivatives of carbohydrates
... developing new drugs: (i) synthesis of analogues of existing drugs; and (ii) search for novel structures that the bacteria have never been presented to before 12 ...the synthesis of a ... See full document
7
Design synthesis and biological evaluation of new antiplasmodial compounds related to ellagic acid
... chloroquine and mefloquine, and it shows no toxicity on human cells at 100 ...vivo studies, synergistic activities with chloroquine, mefloquine, artesunate and atovaquone, and it ... See full document
41
Synthesis and biological evaluation of new 2-benzylchromones
... their studies in the possibility of combine scutellarein, a chromone with numerous pharmacological properties related to neurological disorders, with Rivastigmine, a carbamate compound actually used as AChE ... See full document
123
Phthalocyanine-sulfonamide conjugates-synthesis and biological activity
... effect on two cancer cell lines - human colon (DLD-1) and lung (A549) carcinoma ...2 and subcellular localization was determined by fluorescence ...alone and combination of light was ... See full document
206
Antitumor chalcone derivatives: synthesis and biological activity evaluation
... stirring and on ice. Then, a solution of appropriately substituted benzaldehyde ...h, and was monitored by ...ice and the pH was adjusted to approximately 7 with diluted hydrochloride ... See full document
117
Synthesis, characterization and catalytic studies of new Mo(II)and W(II) complexes and new supporting materials
... distances and angles are given in Table ...ligand and the two carbons from the carbonyl groups determining a fac arrangement (as explained before for the similar structure of ...Mo-N(11) and Mo-N(18) ... See full document
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