[PDF] Top 20 Synthesis and antimicrobial activities of 5arylidenethiazolidine2,4dione derivatives
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Synthesis and antimicrobial activities of 5arylidenethiazolidine2,4dione derivatives
... inactivation of the drug, prevention of the penetration of the target site within the microbe, and alteration of drug target ...development of new derivatives to be used ... See full document
9
Synthesis and antimicrobial, antifungal and anthelmintic activities of 3H-1,5-benzodiazepine derivatives
... active and is directed towards the synthesis of compounds with enhanced pharmacological ...condensation of o-phenylenediamines with α , β -un- saturated carbonyl compounds, 5 β -haloketones or ... See full document
7
Synthesis, Characterization and antimicrobial activity of Cyanopyridine derivatives with Vanillin.
... range of therapeutic activities. Most derivatives are prepared by manipulation of pyridine and its simple homologues in a manner similar to chemistry of the benzenoid ... See full document
5
Synthesis and antimicrobial activity of new amino derivatives of pyrano[4’’,3’’:4’,5’]pyrido[3’,2’:4,5]thieno[3,2-d]pyrimidine
... thienopyrimidine derivatives attracted big interest of the scientific community due to their broad spectrum of biological activities among which are the inhibition of phosphodiesterase, ... See full document
15
SYNTHESIS AND ANTIMICROBIAL ACTIVITIES OF NEW PYRAZOLOPYRIDAZINE DERIVATIVES
... field of medicinal chemistry. Pyridazine ring is a part of the structures of a number of drugs available in the market 1 like cadralazine, minaprine, hydralazine, pipofezine, etc (Figure ... See full document
7
Synthesis and Anti-Mycobacterium tuberculosis Evaluation of Aza-Stilbene Derivatives
... one of the leading causes of death in the world, reaching a million deaths ...2007 and 456,000 deaths among individuals infected with both TB and ...TB, and TB/HIV are stifling attempts ... See full document
8
Synthesis and Antibacterial Evaluation of 3,5-Diaryl-1,2,4-oxadiazole Derivatives
... the synthesis of twenty 3,5-diaryl-1,2,4-oxadiazole derivatives, nine of which are novel ...mirabilis and Staphylococcus ...(MIC) of the active compounds were determined by ... See full document
12
Docking, synthesis and activity of Nacylhydrazone derivatives designed as A4 analogues
... protein, and the results were compared to the data obtained with CA4 (Table ...5m and 5n) were predicted to display better binding than ...5m and 5n display complementary interactions using the ... See full document
16
Synthesis and antitubercular evaluation of new 1,2,3-triazole derivatives of carbohydrates
... preparation of novel 1,4-disubstituted-1,2,3-triazoles derivatives from D- glucose and D-fructose and their in vitro antibacterial activity against Mycobacterium tuberculosis were ...chemical ... See full document
7
Synthesis and biological evaluation of mono and bis-naphthalimide derivatives against SH-SY5Y, human brain cancer cells
... mono and bis-naphthalimides interact with the DNA, was carried out according to the following experiment: a 200 µM de SSC Buffer was prepared mixing 250 µL of x 20 SSC Buffer in 475 mL of distillated ... See full document
169
The antimicrobial activity of lapachol and its thiosemicarbazone and semicarbazone derivatives
... version of the protocol previously described by Gazzinelli et ...matology and Haemotherapy Centre Foundation (proto- col ...volunteers of both sexes by the centrifugation of heparinised venous ... See full document
10
1,2,4-triazine derivatives: Synthesis and biological applications
... panel of six candidate Wnt/ β-catenin/Tcf-regulated genes and found that two of them (Axin2, Lgr5) were reproducibly activated (9–10 fold) in rat intestinal epithelial cells (IEC-6) following ... See full document
14
Antimicrobial, Anti-Inflammatory and Antioxidant Activities of Polyoxygenated Chalcones
... results of the antifungal activity assay using phytopathogens (Table 5) indicate a high sensitivity to the chalcones, with growth inhibition percentages higher than 51%, at all concentrations ...growth of ... See full document
19
Synthesis and evaluation of the phytotoxic activity of α-Santonin derivatives.
... SYNTHESIS AND EVALUATION OF THE PHYTOTOXIC ACTIVITY OF α-SANTONIN ...Mixtures of α-Santonin and various solvents were irradiated by either high or low pressure mercury ...(32%) ... See full document
6
Evaluation of bioactivities of a propolis sample (Gerês) of Portuguese origin
... choice of the yeast ...non-pathogenicity, and the well- known biology, genetics and metabolism (Guthrie and Fink, ...stages of growth. After a short period of adjustment, the lag ... See full document
96
Synthesis, Anti-Inflammatory and Anti- Nociceptive Activities and Cytotoxic Effect of Novel Thiazolidin-4-ones Derivatives as Selective Cyclooxygenase (COX-2) Inhibitors
... structure of protein was downloaded from protein data bank (PDB ID: 1cx2) and further preparations like removing water molecules and adding polar hydrogens were done using AutoDock tools ...software ... See full document
7
Anti-Parasite and Cytotoxic Activities of Chloro and Bromo L-Tyrosine Derivatives
... strains of medical importance as Candida tropicalis (ATCC 750), ...isolates and strains of filamentous fungi were included: Sporothrix schenckii (UdeA 7027), ...24198) and Fusarium oxysporum ... See full document
11
Urease inhibitory activities of beta-boswellic acid derivatives
... concentrated and solvent was ...fraction and ex- traction was performed by ethyl acetate five ...2%, and previous step was ...related derivatives in organic ...filtered and concentrated ... See full document
6
One pot synthesis of 2-hydroxy pyrrolidine derivatives
... utility of domino reaction between aryl amines, in particularly with various anilines and cyclic enol ethers such as 2,3-dihydrofuran and 3,4-dihydro-2H-pyran in the straight forward synthesis ... See full document
6
Synthesis, characterization and antifungal activity of quaternary derivatives of chitosan on Aspergillus flavus
... tion of chitin, which after cellulose is the second most abundant natural biopolymer found in ...exoskeletons of arthropods of crustaceans, fungi, insects, annelids, mollusks and coelenter- ... See full document
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